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Antagonis Kolinergik Antagonis Adrenergik

This document lists various classes of drugs and examples of drugs within each class. It covers drugs that act on the autonomic nervous system, central nervous system, cardiovascular system, and others. The classes include adrenergic agonists and antagonists, cholinergic agonists and antagonists, benzodiazepines, anesthetics, antihypertensives, diuretics, and many others.

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0% found this document useful (0 votes)
128 views

Antagonis Kolinergik Antagonis Adrenergik

This document lists various classes of drugs and examples of drugs within each class. It covers drugs that act on the autonomic nervous system, central nervous system, cardiovascular system, and others. The classes include adrenergic agonists and antagonists, cholinergic agonists and antagonists, benzodiazepines, anesthetics, antihypertensives, diuretics, and many others.

Uploaded by

marsella
Copyright
© © All Rights Reserved
Available Formats
Download as DOCX, PDF, TXT or read online on Scribd
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ANTAGONIS ADRENERGIK ANTAGONIS KOLINERGIK

PENGHAMBAT -α PELEMAS
OBAT ANTIMUSKARINIK
- Alfuzosin - Prazosin NEUROMUSKULAR
- Doxazosin - Tamsulosin
Atropine
- Phenoxybenzamine - Terazosin
- Phentolamine - Yohimbine Cyclopentolate Atracurium
Ipratropium Cisatracurium
PENGHAMBAT -β
Scopolamine Doxacurium
- Acebutolol - Metoprolol Tropicamide Metocurine
- Atenolol - Nadolol
PENGHAMBAT Mivacurium
- Carvedilol - Pindolol
GANGLIONIK Pancuronium
- Esmolol - Propanolol
- Labetalol - Tomolol Rocuronium
Succinylcholine
OBAT YANG MEMENGARUHI PELEPASAN ATAU Mecamylamine
Tubocurarin
PENGAMBILAN KEMBALI NEUROSTRANSMITER Nicotine
Vecuronium
- Guanethidine - Reserpine

AGONIS KOLINERGIK AGONIS ADRENERGIK

KERJA LANGSUNG KERJA LANGSUNG


KERJA TAK LANGSUNG
(reversibel)
Asetilkolin - Albuterol - Metaproterenol
Bethanechol - Clonidine - Methoxamine
Carbachol Ambenomium - Dobutamine - Norepinephrine
Cevimeline - Dopamine - Phenylephrine
Demecarium
Pilocarpine - Epinephrine - Pirbuterol
Donezepil - Formoterol - Salmeterol
KERJA TAK LANGSUNG
Edrophonium - Isoproterenol - Terbutaline
(ireversibel) Galantamine
Neostigmine KERJA TIDAK LANGSUNG
Echothiophate Physostigmine
Pyridostigmine - Amphetamine - Tyramine - Cocaine
REAKTIVASI ASETIL
KOLIN ESTERASE Rivastigmine KERJA LANGSUNG & TIDAK LANGSUNG
Tacrine (KERJA CAMPURAN)

Pralidoxime - Ephedrine - Pseudoephedrine


BENZODIAZEPINE OBAT-OBAT ANTI PARKINSON
- Alprazolam - Flurazepam
- Amantadine - Pramipexole
- Chlordiazepoxide - Lorazepam - Apomorphine - Procyclidine
- Clonazepam - Quazepam - Benztropine - Rasagiline
- Clorazepate - Oxazepam - Biperiden - Ropinirole
- Diazepame - Temazepame - Bromocriptine - Rotigotine
- Estazolam - Triazolam - Carbidopa - Selegiline (Deprenyl)
- Entacapone - Talcapone
ANTAGONIS BENZODIAZEPINE - Levodopa - Trihexypenidyl

- Flumazenil OBAT-OBAT ANTI ALZHEIMER

OBAT-OBAT ANXIOLITIK LAIN - Donepezil - Rivastigmine


- Buspirone - Antidepresan - Galantamine - Tacrine
- Hydroxyzine - Memantine

BARBITURAT
- Amobarbital - Secobarbital
- Phenobarbital - Thiopental
- Pentobarbital PERANGSANG PSIKOMOTOR

OBAT HIPNOTIK LAINNYA - Amphetamine - Methylphenidate


- Armodafinil - Modafinil
- Antihistamin - Ramelteon
- Atomoxentine - Nicotine
- Chloral hydrate - Zalepion
- Caffeine - Theobromine
- Eszopicion - Zolpidem
- Cocaine - Teophylline
- Ethanol
- Dextroamphetamine - Varenicline
- Lisdexamphetamine

HALUSINOGEN

- Lysergic acid diethylamide (LSD)


- Phencyclidine (PCP)
- Tetrahydrocannabinol (THC)
OBAT-OBAT PRANESTETIK PENGHAMBAT AMBILAN-KEMBALI
- Antikolinergik - Benzodiazepin SEROTONIN SELEKTIF
- Antiemetik - Pelemas otot - Citalopram - Fluvoxamine
- Antihistamin - Oploid - Escitalopram - Paroxetine
- Barbiturat - Fluoxetin - Sertraline

ANESTETIK UMUM PENGHAMBAT AMBILAN-KEMBALI


NOREPINEFRIN/SEROTONIN
INHALASI INTRAVENA
- Duloxetine - Venlafaxine
- Desflurane - Barbiturat
- Enflurane - Benzodiazepine ANTIDEPRESAN ATIPIKAL
- Halothane - Etomidate
- Isoflurane - Ketamine - Bupropion - Nefazodone
- Nitrous Oxide - Oploid - Mirtazapine - Trazodone
- Sevoflurane - Propofol
ANTIDEPRESAN TRISIKLIK
ANESTETIK LOKAL
- Amitriptyline - Imipramine
- Bupivacaine - Procaine - Amoxapine - Maprotiline
- Lidocaine - Tetracaine - Clomipramine - Nortriptyline
- Desipramine - Protriptyline
- Doxepine - Trimipramine

PENGHAMBAT MONOAMINA OKSIDASE


OBAT-OBAT ANTIEPILEPTIK - Phenelzine - Tranylcypromine
- Selegiline
- Barbiturat - Levetiracetam
- Benzodiazepine - Oxcarbazepine OBAT-OBAT YANG DIGUNAKAN UNTUK MENGOBATI
- Carbamazepine - Phenytoin MANIA DAN GANGGUAN BIPOLAR
- Divalproex - Pregabalin
- Ethosuximide - Primidone - Carbamazepine - Valproic acid
- Felbamate - Tiagabine - Garam lithium
- Gabapentine - Topiramate
- Lamotrigine - Zonisamide
AGONIS KUAT NEUROLEPTIK TIPIKAL (potensi rendah)

- Alfentanil - Morphine
- Fentanyl - Oxycodone - Chlorpromazine - Thioridazine
- Heroin - Remifentanil - Prochlorperazine
- Meperidine - Sufentanil
- Methadone NEUROLEPTIK TIPIKAL (potensi tinggi)

AGONIS SEDANG/LEMAH
Codeine - Fluphenazine - Pimozide
- Codeine - Propoxyphene - Haloperidol - Thiothixene
ANTAGONIS – AGONIS CAMPURAN DAN
NEUROLEPTIK ATIPIKAL
AGONIS PARSIAL
- Buprenorphine - Nalbuphine - Aripriprazole - Paliperidone
- Butorphanol - Pentazocine - Chlozapine - Risperidone
ANTAGONIS - Olanzapine - Ziprasidone
- Quetiapine
- Nalmefene - Naltrexone
- Naloxone
ANALGESIK LAIN OBAT OBAT DIURETIK
- Tramadol DIURETIK TIAZID

ANGINA - Chlorothiazide - Indapamide


(OBAT-OBAT ANTIANGINA) - Chlorthalidone - Metolazone
- Hydrochlorothiazide
NITRAT ORGANIK
LOOP DIURETIC
- Isosorbide dinitrate
- Bumetanide - Furosemide
- Isosorbide mononitrate
- Ethacrynic acid - Torsemide
- Nytroglycerin
DIURETIK HEMAT - KALIUM
PENGHAMBAT –β
- - Acebutolol - Metoprolol - Amiloride - Spironolactone
- Atenolol - Propanolol - Eplerenone - Triamteren

PENGHAMBAT KANAL Ca 2+ PENGHAMBAT KARBONIK ANHIDRASE

- Amlodipine - Nicardipine - Asetazolamid


- Diltiazem - Nifedipine DIURETIK OSMOTIK
- Felodipine - Verapamil - Mannitol - Urea
HIPERTENSI
GAGAL JANTUNG (OBAT-OBAT ANTIHIPERTENSI)
(OBAT-OBAT YANG DIGUNAKAN UNTUK MENGOBATI
GAGAL JANTUNG) DIURETIK
PENGHAMBAT SISTEM RENIN ANGIOTENSI. - Bumetanide - Hydrochlorothiazide
- Eplerenone - Spironolacton
PENGHAMBAT PENGHAMBAT RESEPTOR - Furosemide - Triamterene
ACE ANGIOTENSIN
PENGHAMBAT –β
- Captopril
- Enalapril - Candesartan - Atenolol - Nadolol
- Fosinopril - Losartan - Carvedilol - Propranolol
- Lisinopril - Telmisartan - Labetalol - Timolol
- Quinapril - Valsartan - Metoprolol
- Ramipril PENGHAMBAT ACE
PENGHAMBAT –β - Benazepril - Lisinopril
- Atenolol - Metoprolol - Captropil - Moexipril
- Carvedilol - Enalapril - Quinapril
- Fosinopril - Ramipril
DIURETIK
ANTAGONIS RESEPTOR ANGIOTENSIN II
- Bumetanide - Hydrochlorothiazide
- Furosemide - Metolazone - Candesartan - Olmesartan
- Eprosartan - Telmisartan
VASODILATOR LANGSUNG - Irbesartan - Valsartan
- Losartan
- Hydralazine
PENGHAMBAT RENIN
- Isosorbide dinitrate
- Sodium nitroprusside - Aliskiren

AGEN INOTROPIK PENGHAMBAT KANAL Ca2+


- Amrinone - Dobutamine - Amlodipine - Nicardipine
- Diltiazem - Nifedipine
- Digitoxin - Mirinone
- Felodipine - Nisoldipine
- Digoxin - Isradipine - Verapamil
ANTAGONIS ALDOSTERON PENGHAMBAT - α
- Spironolacton - Doxazosin - Terazosin
- Prazosan
LAIN - LAIN
- Clonidine - α methyldopa
- Diazoxide - Minoxidil
- Hydralazine - Sodium Altropruside
- Labetalol
ARITMA
(OBAT-OBAT ANTIARITMA)
KELAS I (Penghambat kanal Na+) PENGHAMBAT HMG KoA REDUKTASE
- Dysopiramide (IA) - Procainamide (IA) - Atorvastatin - Pravastatin
- Flecainide (IC) - Propafenone (IC) - Fluvastatin - Rosuvastatin
- Lidocaine (IB) - Quinidine (IA) - Lovastatin - Simvastatin
- Mexlletine (IB) - Tocainide (IB)

KELAS II (Penghambat adrenoreseptor –β)


- Fenofibrate - Gemfibrozil
- Esmolol - Propranolol
- Metoprolol
KELAS III (Penghambat kanal K+)
- Amiodarone - Sotalol - Colesevelam - Cholestyramine
- Dofetilide - Colestipol
KELAS IV (Penghambat kanal Ca+)

- Diltiazem - Verapamil
- Ezetimibe
OBAT-OBAT ANTIARITMA LAINNYA

- Adenosine - Digoxin OBAT-OBAT ANTI-INFLAMASI

HIPOLIPIDEMIK OAINS
ASAM FIBRAT - Aspirin - Meloxicam
- Bezafibrat - Klofibrat - Diflunisal - Methyl Salicylate
- Fenofibrat - Siprofibrat - Diclofenac - Nabumetone
- Gemfibrozil - Etodolac - Naproxen
- Fenamate - Oxaprozin
RESIN - Flurbiprofe - Piroxicam
- Kelesteramin - Kolestipol - Ibuprofen - Sulindac
PENGHAMBAT HMG-CoA REDUKTASE - Indomethacin - Tolmetin
- Ketoprofen - Ketorolac
- Lovastatin - Pravastatin
- Mevastatin - Simvastatin PENGHAMBAT COX- 2
ASAM NIKOTINAT
- Celecoxib
- Asam Nicotinat - Asipimoks
ANALGESIK LAINNYA
LAIN-LAIN
- Bekatul -Neosimin sulfat - Acetaminophen
- Betasitosterol - Probukol
- Dekstrotirosin
- Abciximab - Eptifibatide
- Aspirin - Ticlopidine
- Clopidogrel - Tirofiban
- Dipyridamole

- Argatroban - Heparin
- Dalteparin - Lepirudin
- Enoxaparine - Warfarin
- Fondaparinus

- Altepiase (tPA) - Streptokinase

- Aminocaproic acid - Tranexamic acid


- Aprotinin - Vitamin K
- Protamine sulfate

- Cyanocobalamin (B12) - Folic acid


- Erythropoietin - Besi

- Hydroxyurea
OBAT-OBAT ANTI-INFLAMASI

OAINS

- Aspirin - Meloxicam
- Diflunisal - Methyl Salicylate
- Diclofenac - Nabumetone
- Etodolac - Naproxen
- Fenamate - Oxaprozin
- Flurbiprofe - Piroxicam
- Ibuprofen - Sulindac
- Indomethacin - Tolmetin
- Ketoprofen - Ketorolac

PENGHAMBAT COX- 2
- Celecoxib

ANALGESIK LAINNYA
- Acetaminophen

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